pKa | 6.6 |
---|---|
Half-life | Â |
Route oral | 4 h (range 1–14) |
Intramuscular | 12 h (range 8–23) |
Inhalatory route | 4 h (range 6–8) |
Time to peak concentration | Â |
Route oral | 1 h |
Intramuscular | 5 h |
Inhalatory route | 2 min (1–3) |
Metabolites | 7- and 8-Hydroxyloxapine |
Desmethyl-loxapine (amoxapine) | |
7- and 8-Hydroxyamoxapine | |
 | Ioxapine N-oxide |
Excretion | Excretion of glucuronide conjugates in urine |
Unchanged in faeces |